Isakhiwo samangqamuzana:
I-Cytisine yenzeka ngokwemvelo i-alkaloid etholakala ezinhlotsheni zezitshalo eziningana, njengeCytisus ashoninum kanye ne-labingburm anagyroides. Kusetshenziswe iminyaka eminingi njengosizo lwenkohliso yokubhema ngenxa yokufana kwayo ku-nicotine.Umsebenzi oyinhloko we-cytisine unjenge-ageptors engxenye ye-nicotinic acetylcholine (NACHRS). Lezi receptors zitholakala ebuchosheni, ikakhulukazi ezindaweni ezibandakanyeka ekuthathweni, futhi banesibopho sokulalela imiphumela enomvuzo ye-nicotine. Ngokubopha futhi kusebenze le receptors, i-cytisine kusiza ukunciphisa izifiso ze-nicotine kanye nezimpawu zokuhoxisa ngesikhathi sokubhema Kungasiza ukuthuthukisa amanani okuyeka futhi kunciphise ubukhulu bezimpawu zokuhoxisa, okwenza kube lusizo oluwusizo ekubhemeni izinhlelo zokucacisa.
Kubalulekile ukuqaphela ukuthi i-cytisine ingaba nemiphumela emibi, efana ne-nausea, ukugabha, nokuphazamiseka kokulala. Njenganoma imuphi umuthi, kufanele isetshenziswe njengoba kuqondiswe futhi ngaphansi kokugadwa kochwepheshe wezokunakekelwa kwempilo. Uma ucubungula usebenzisa i-cytisine njengosizo lokuphuthuma lwenkohliso, ngincoma ukubonisana nodokotela wakho ngeseluleko nesiqondiso sabantu.
Into yendaba | Ukucacisa | |
Assay (HPLC) | ||
I-Cytisine: | ≥98% | |
Okujwayelekile: | I-CP2010 | |
-Obukhali | ||
Ukubukeka: | I-Light Yellow Crystalline Powder | |
Iphunga: | Umphumo wengqondo | |
Inqwaba density: | I-50-60g / 100ml | |
Mesh: | 95% udlule 80mesh | |
Metal esindayo: | ≤10pppm | |
Njengo: | ≤2ppm | |
PB: | ≤2ppm | |
Ukulahlekelwa ukoma: | ≤1% | |
I-Specid Resed: | ≤0.1% | |
Insalela ye-solvent: | ≤3000ppp |